LI Xuqin
(2) Design, synthesis of small molecules as biomedical agents
Prof. Xuqin Li obtained her B.S. from Lanzhou University in 1999 and M.S with Prof. Zhongjian Jia in 2002. After that, she pursued her Ph.D. from the Institute of Materia Medica, Chinese Academy of Medical Science with Prof. Gang Liu (2002-2005). From 2005 to 2007, she worked as a research associate with Prof. Burkhard Koenig in University of Regensburg, Germany, and with Prof. Malcolm Stevens, Pharminox Ltd., Nottingham, United Kingdom. In 2007, she started her independent career as a lecture in the Department of Chemistry, University of Science and Technology Beijing, and was promoted to an associate professor in 2011. Her research interests mainly focus on synthetic organic chemistry and medicinal chemistry.
(1) The preparation and application of Anthranilic acid derivatives. Xuqin Li, Chi-Hin Cho, Kenneth K.W. To,Kai Zheng, Lin Wang, Yan Lei, Yangyang Zhao. Faming Zhuanli Shenqing (2014), CN 201410772734.1.
Patent:
(1) The preparation and application of Anthranilic acid derivatives. Xuqin Li, Chi-Hin Cho, Kenneth K.W. To,Kai Zheng, Lin Wang, Yan Lei, Yangyang Zhao. Faming Zhuanli Shenqing (2014), CN 201410772734.1.
(2) Xuqin Li, An Liu, Feilong Zhang, Yan Lei, “The preparation and application of Anthranilic acid derivatives”, Faming Zhuanli Shenqing (2012), CN 201210063762.7.
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(1) Huu-Manh Vu, Jia-Yuan Yong, Fei-Wu Chen, Xu-Qin Li,* and Guo-Qing Shi, Rhodium-Catalyzed C(sp2)-H Amidation of Azine with Sulfonamides, J. Org. Chem. 2020, 85, 4963-4972. DOI: 10.1021/acs.joc.0c00138 (SCI, Top)
(2) Jia-Yuan Yong; Huu-Manh Vu; Xu-Qin Li;* Ai-Jun Gong, Palladium (0)-catalyzed C(sp2)-H oxygenation with carboxylic acids, Tetrahedron, 2020, 76(10), DOI: 10.1016/j.tet.2020.130969 (SCI)
(3) Huu Manh Vu, Fei-Wu Chen, Xu-Qin Li,* Acetoxylation and Halogenation of 2-arylbenzoxazinones via Palladium-Catalyzed C(sp2)-H Bond Oxidation, Chemistryselect, 2019, 4(32), 9465-9469. DOI: 10.1002/slct.201902611 (SCI)
(4) Vu, Huu-Manh; Li, Xu-Qin;* Chen, Fei-Wu, Palladium-Catalyzed C-H Bond Monofluorination of 2-Arylbenzo[d]oxazinone Using Nitrate as Crucial Promoter, Synthesis, 2019, 51(7), 1578-1584. DOI: 10.1055/s-0037-1611700 (SCI)
(5) Xianxing Shang, Huu-Manh Vu, Xuqin Li*, One-Pot Synthesis of 2-Arylbenzoxazinones from 2-Arylindoles with (Diacetoxyiodo)benzene as the Sole Oxidant, Synthesis, 2018, 50(2), 377-383. DOI: 10.1055/s-0036-1590933 (SCI)
(6) Hanrui Yang, Jiejie Wang, Pengpeng Shao, Siyi Yuan, Xuqin Li*, A facile three-step total synthesis of tanshinone I, J. Asian Nat. Prod. Res., 2016, 18(7), 677-683. DOI: 10.1080/10286020.2015.1136906 (SCI)
(7) Xuqin Li*, Lin Wang, Yan Lei, Tao Hu, Fei-Long Zhang, Chi-Hin Cho, Kenneth K.W. To*, Reversal of P-gp and BCRP-mediated MDR by Tariquidar derivatives, Eur. J. Med. Chem., 2015, 101, 560-572. DOI: 10.1016/j.ejmech.2015.06.049 (SCI)
(8)Tao Ban, Huu-Manh Vu, Jing Zhang, Jia-Yuan Yong, Qiong Liu, and Xu-Qin Li*, Rhodium-Catalyzed Azine-Directed C–H Amidation with N-Methoxyamides, J. Org. Chem., 87, 5543-5555. DOI: 10.1021/acs.joc.1c02868 (2022)
(9)Qiong Liu, Jia-Yuan Yong, Jing Zhang, Tao Ban, Xu-Qin Li*, C-H acylation of Aniline derivatives with α-Oxocarboxylic Acids under Ruthenium Catalyst, Org. Biomol. Chem., DOI: 10.1039/D2OB01212J (2022)
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